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hERG
Gene: KCNH2
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Standard throughput time | 2 weeks |
Source | human | |
Expression system | mammalian (CHO, HEK 293), stable expression | |
Method | manual and automated patch-clamping | |
Quality level | high quality functional assay | |
References | E-4031 | |
Further References | Dofetilide, Terfenadine, Ketoconazole | |
Additional readouts | solubility check, stability check | |
+ Should be used for quality characterization of hERG interaction | ||
+ IKr screen |