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KVLQT1/minK
Cell lines available: HEK293 / CHO, constitutive expression. Assays validated for manual and automated patch-clamp.
Manual patch-clamp:
|
IC50 value (µM) |
|
IC50 value (µM) |
Chromanol |
6.2 |
Mefloquine |
3.6 |
Automated patch-clamp:
|
IC50 value (µM) |
Mefloquine |
12.3 |