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KV4.3 (IKto)
Cell lines available: CHO, constitutive expression. Assays validated for manual and automated patch-clamp.
Manual patch-clamp:
|
IC50 value (µM) |
|
IC50 value (µM) |
Dapoxetine HCl |
12.4 |
Dapoxetine HCl |
3.0 |
Automated patch-clamp :
|
IC50 value (µM) |
Dapoxetine HCl instantaneous |
46.3 |